LCB

Publications de l’année 2008

1. Umpolung reactivity of difluoroenol silyl ethers with amines and amino alcohols. Application to the synthesis of enantiopure alfa-difluoromethyl amines and amino acids, Huguenot, F. ; Billac, A. ; Brigaud, T. ; Portella, C. J. Org. Chem. 2008, 73, 2564-2569

2. Concise access to enantiopure (S)- and (R)-α-trifluoromethyl pyroglutamic acids from ethyl trifluoropyruvate-based chiral CF3-oxazolidines (Fox), Chaume, G. ; Van Severen, M. -C. ; Ricard, L. ; Brigaud, T. J. Fluorine Chem. 2008, 129, 1104-1109

3. Fluorine••• and π•••Alcali Metal Interactions control in the Stereoselective Amide Enolates Alkylation using Fluorinated Oxazolidines (Fox) as Chiral Auxiliary : An Experimental and Theoretical Study, Sini, G. ; Tessier, A. ; Pytkowicz, J. ; Brigaud, T. Chem. Eur. J. 2008, 14, 3363-3370

4. Highly diastereoselective synthetic route to enantiopure β2-amino acids and γ-amino alcohols using a fluorinated oxazolidine (Fox) as chiral auxiliary, Tessier, A. ; Lahmar, N. ; Pytkowicz, J. ; Brigaud, T. J. Org. Chem. 2008, 73, 3970-3973

5. Direct C-glycosylation by indium-mediated alkynylation on sugar anomeric position, Lubin-Germain, N. ; Baltaze, J. -P. ; Coste, A. ; Hallonet, A. ; Lauréano, H. ; Legrave, G. ; Uziel, J. ; Augé, J. Org. Lett. 2008, 10, 725-728

6. Synthesis of P-stereogenic phosphorus compounds based on chiral aminoalcohols as chiral auxiliary, Darcel, C. ; Uziel, J. ; Juge, S. Phosphorus Ligands in Asymmetric Catalysis 2008, 3, 1211-1233.

7. A new rationale of reaction metrics for green chemistry. Mathematical expression of the environmental impact chemical processes, Augé, J. Green Chem. 2008, 10, 225-231

8. Novel sst5-Selective Somatostatin Dicarba-Analogues : Synthesis and Conformation-Affinity Relationships, D’Addona, D. ; Carotenuto, A. ; Novellino, E. ; Piccand, V. ; Reubi, J. C. ; Di Cianni, A. ; Gori, F. ; Papini, A. M., Ginanneschi, M. J. Med. Chem. 2008, 51, 512-520

9. Ferrocenyl Glycopeptides as Electrochemical Probes to Detect Autoantibodies in Multiple Sclerosis Patients’ Sera, Real Fernández, F. ; Chamois-Colson, A. ; Bayardon, J. ; Nuti, F. ; Peroni, E. ; Meunier-Prest, R. ; Lolli, F. ; Chelli, M. ; Darcel, C. ; Jugé, S. ; Papini, A. M. Pept. Science 2008, 90, 488-495

10. Synthesis and Conformational Analysis of a Cyclic Peptide Obtained via i to i+4 Intramolecular Side-Chain-to-Side-Chain Azide-Alkyne 1,3-Dipolar Cycloaddition, Cantel, S. ; Le Chevalier-Isaad, A. ; Scrima, M. ; Levy, J. J. ; DiMarchi, R. D. ; Rovero, P. ; Halperin, J. A. ; D’Ursi, A. M. ; Papini, A. M. ; Chorev, M. J. Org. Chem. 2008, 73, 5663-5665

11. Design glycopeptides with different β-turn types as synthetic probes for the detection of autoantibodies of multiple sclerosis, Carotenuto, A. ; Alcaro, A. C. ; Saviello, M. R. ; Peroni, E. ; Nuti, F. ; Papini, A. M. ; Novellino, E. ; Rovero, P. J. Med. Chem. 2008, 51, 5304-5309

12. Optimized strategies for the synthesis of biomolecules by the microwave approach Paolini, I. ; Rizzolo, F. ; Papini, A. M. Chem. Today 2008, 26(Supl), 36-38

13. N-α-Fmoc-protected ω-azido and ω-alkynyl-L-aminoacids as building blocks for the synthesis of “clickage” peptides, Le Chevalier Isaad, A. ; Barbetti, F. ; Rovero, P. ; D’Ursi, A. M. ; Chelli, M. ; Chorev, M. ; Papini, A. M. Eur. J. Org. Chem. 2008, 5308-5314

14. Advances in automatic, manual and microwave-assisted solid-phase peptide synthesis, Sabatino, G. ; Papini, A. M. Curr. Opin. Drug Discov. Devel. 2008, 11, 762-770

15. Ferrocenyl glycopeptides as electrochemical probes to detect autoantibodies in multiple sclerosis patients’ sera, Real-Fernandez, F. ; Colson, A. ; Bayardon, J. ; Nuti, F. ; Peroni, E. ; Meunier-Prest, R. ; Lolli, F. ; Chelli, M. ; Darcel, C. ; Juge, S. ; Papini, A. M. Biopolymers 2008, 90, 488-495